Items where Author is "Cominetti, Marco M D"

Article

Hamshaw, Isabel ORCID: https://orcid.org/0000-0001-6445-0738, Cominetti, Marco, Nana-Akyin, Princess, Ho Yee Ho, Ernie, Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 and Mueller, Anja ORCID: https://orcid.org/0000-0003-0774-0434 (2024) IS4-FAM, a fluorescent tool to study CXCR4 affinity and competitive antagonism in native cancer cells. Pharmacology Research and Perspectives, 12 (5). ISSN 2052-1707

Hayward, Deanne, Goddard, Zoë R. ORCID: https://orcid.org/0000-0002-7900-1553, Cominetti, Marco M. D., Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 and Beekman, Andrew M. ORCID: https://orcid.org/0000-0002-3056-6406 (2024) Light-activated azobenzene peptide inhibitor of the PD-1/PD-L1 interaction. Chemical Communications, 60 (63). pp. 8228-8231. ISSN 1359-7345

Cominetti, Marco M. D., Goddard, Zoë R. ORCID: https://orcid.org/0000-0002-7900-1553, Hood, Bethany R., Beekman, Andrew M. ORCID: https://orcid.org/0000-0002-3056-6406, O'Connell, Maria A. ORCID: https://orcid.org/0000-0002-0267-0951 and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2024) Borylation via iridium catalysed C–H activation: a new concise route to duocarmycin derivatives. Organic & Biomolecular Chemistry, 22 (27). pp. 5603-5607. ISSN 1477-0520

Hamshaw, Isabel ORCID: https://orcid.org/0000-0001-6445-0738, Cominetti, Marco M. D., Lai, Wing-Yee, Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 and Mueller, Anja ORCID: https://orcid.org/0000-0003-0774-0434 (2023) The development of potent, competitive CXCR4 antagonists for the prevention of cancer metastasis. Biochemical Pharmacology, 218. ISSN 0006-2952

Ivens, Eleanor, Cominetti, Marco M. D. and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2022) Junctions in DNA: underexplored targets for therapeutic intervention. Bioorganic & Medicinal Chemistry, 69. ISSN 0968-0896

Bidula, Stefan ORCID: https://orcid.org/0000-0002-3790-7138, Nadzirin, Izzuddin Bin, Cominetti, Marco, Hickey, Harry, Cullum, Sean A., Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949, Schmid, Ralf and Fountain, Samuel J. ORCID: https://orcid.org/0000-0002-6028-0548 (2022) Structural basis of the negative allosteric modulation of 5-BDBD at human P2X4 receptors. Molecular Pharmacology, 101 (1). pp. 33-44. ISSN 1521-0111

M. M. D. Cominetti, Marco, Goddard, Zoë R. ORCID: https://orcid.org/0000-0002-7900-1553, Howman, Chloe E., O'Connell, Maria A. ORCID: https://orcid.org/0000-0002-0267-0951 and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2021) Amino DSA analogues as payloads for antibody-drug conjugates with multiple sites for conjugation. Initial studies and solid phase synthesis. Tetrahedron Letters, 72. ISSN 0040-4039

Goddard, Zoë Rachael ORCID: https://orcid.org/0000-0002-7900-1553, Beekman, Andrew Michael ORCID: https://orcid.org/0000-0002-3056-6406, Cominetti, Marco M. D., O'Connell, Maria A. ORCID: https://orcid.org/0000-0002-0267-0951, Chambrier, Isabelle, Cook, Michael J., Marin, Maria J. ORCID: https://orcid.org/0000-0001-8021-5498, Russell, David A. and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2021) Peptide directed phthalocyanine-gold nanoparticles for selective photodynamic therapy of EGFR overexpressing cancers. RSC Medicinal Chemistry, 12 (2). pp. 288-292. ISSN 2632-8682

Cartwright, Oliver Charles, Beekman, Andrew Michael ORCID: https://orcid.org/0000-0002-3056-6406, Cominetti, Marco M. D., Russell, David A. and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2020) A peptide-duocarmycin conjugate targeting the Thomsen-Friedenreich antigen has potent and selective antitumour activity. Bioconjugate Chemistry, 31 (7). 1745–1749. ISSN 1043-1802

Beekman, Andrew ORCID: https://orcid.org/0000-0002-3056-6406, Cominetti, Marco, Cartwright, Oliver, Boger, Dale L. and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2019) A small molecule drug conjugate (SMDC) of DUPA and a duocarmycin built on the solid phase. MedChemComm, 10 (12). pp. 2170-2174. ISSN 2040-2503

Beekman, Andrew M. ORCID: https://orcid.org/0000-0002-3056-6406, Cominetti, Marco M. D., Walpole, Samuel J., Prabhu, Saurabh, O'Connell, Maria A. ORCID: https://orcid.org/0000-0002-0267-0951, Angulo Alvarez, Jesus ORCID: https://orcid.org/0000-0001-7250-5639 and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2019) Identification of selective protein-protein interaction inhibitors using efficient in silico peptide-directed ligand design. Chemical Science, 10 (16). pp. 4502-4508. ISSN 2041-6520

Bertrand, Benoît, Fernandez-Cestau, Julio, Angulo, Jesus ORCID: https://orcid.org/0000-0001-7250-5639, Cominetti, Marco M. D., Waller, Zoe A. E., Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949, O'Connell, Maria A. ORCID: https://orcid.org/0000-0002-0267-0951 and Bochmann, Manfred ORCID: https://orcid.org/0000-0001-7736-5428 (2017) Cytotoxicity of pyrazine-based cyclometalated (C^Npz^C)Au(III) carbene complexes: Impact of the nature of the ancillary ligand on the biological properties. Inorganic Chemistry, 56 (10). 5728–5740. ISSN 0020-1669

Cominetti, Marco M. D., Hughes, David L. and Matthews, Susan E. ORCID: https://orcid.org/0000-0001-8821-0851 (2016) Open-resorcinarenes, a new family of multivalent scaffolds. Organic & Biomolecular Chemistry, 14 (43). pp. 10161-10164. ISSN 1477-0520

Cominetti, Marco, Goffin, Sarah, Raffel, Ewan, Turner, Kerrie, Ramoutar, Jordann, O'Connell, Maria ORCID: https://orcid.org/0000-0002-0267-0951, Howell, Lesley and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2015) Identification of a new p53/MDM2 inhibitor motif inspired by studies of chlorofusin. Bioorganic & Medicinal Chemistry Letters, 25 (21). pp. 4878-4880. ISSN 0960-894X

Pergolizzi, Giulia, Cominetti, Marco, Butt, Julea N. ORCID: https://orcid.org/0000-0002-9624-5226, Field, Robert A. ORCID: https://orcid.org/0000-0001-8574-0275, Bowater, Richard ORCID: https://orcid.org/0000-0002-2745-7807 and Wagner, Gerd K. (2015) Base-modified NAD and AMP derivatives and their activity against bacterial DNA ligases. Organic & Biomolecular Chemistry, 13. pp. 6380-6398. ISSN 1477-0520

Book Section

Beekman, Andrew ORCID: https://orcid.org/0000-0002-3056-6406, Cominetti, Marco M D and Searcey, Mark ORCID: https://orcid.org/0000-0003-2273-8949 (2019) Duocarmycins as Antibody–Drug Conjugate (ADC) Payloads. In: Cytotoxic Payloads for Antibody-Drug Conjugates. Royal Society of Chemistry. ISBN 978-1-78801-077-1